T12358 |
Palonidipine
|
96515-73-0
|
98%
|
|
Palonidipine is an antagonist of calcium, is potential for the therapy of angina-pectoris and hypertension.
|
T8199 |
(±)-α-Bisabolol
|
515-69-5
|
98%
|
|
(±)-α-Bisabolol is a natural product from Vanillosmopsis erythropappa
|
TN2641 |
15-Methoxypinusolidic acid
|
769928-72-5
|
98%
|
|
15-Methoxypinusolidic acid has anti-inflammatory effects, it inhibits LPS-induced iNOS expression and NO production, independent on MAPK and NF-kappaB. 15-Methox...
|
T12205L |
Trans-Ned 19
|
1354235-96-3
|
98%
|
|
trans-Ned 19 is a NAADP antagonist and TPC blocker and inhibits the calcium signal in human umbilical vein endothelial cells and the rat aorta relaxation in resp...
|
TL0014 |
Pinusolide
|
31685-80-0
|
98%
|
|
Pinusolide is a platelet activating factor ( PAF) antagonist, it may prove of therapeutic value in the treatment of hypotension, it has antileukemic potential, a...
|
TQ0145 |
(R)-(+)-Bay-K-8644
|
98791-67-4
|
98%
|
|
(R)-(+)-Bay K 8644 is a calcium channel inhibitor. It inhibits Ba2+ currents (IBa) (IC50: 975 nM).
|
TN2169 |
Saikogenin D
|
5573-16-0
|
98%
|
|
Saikogenin D possesses a dual effect: an inhibition of A23187-induced PGE2 production without a direct inhibition of cyclooxygenase activity; and an elevation of...
|
TN5109 |
Taxezopidine L
|
219749-76-5
|
98%
|
|
Taxezopidines K and taxezopidine L can markedly inhibit Ca2+-induced depolymerization of microtubules.
|
T16357 |
NSC 663284
|
383907-43-5
|
98%
|
|
NSC 663284 is a cell-permeable and irreversible Cdc25 dual specificity phosphatase inhibitor (IC50 for Cdc25B2: 0.21 μM). NSC 663284 inhibits NSD2 (IC50 of 170 n...
|
TN2287 |
Turkesterone
|
41451-87-0
|
98%
|
|
Turkesterone is a phytoecdysteroid possessing an 11alpha-hydroxyl group, also is an analogue of the insect steroid hormone 20-hydroxyecdysone. It has immunomodul...
|
T12322 |
ORM-10962
|
763926-98-3
|
98%
|
|
ORM-10962 is a potent, highly selective inhibitor of sodium-calcium exchanger (NCX) (for the reverse and forward mode inhibition with IC50 values of 67 and 55 nM...
|
T13250 |
UK51656
|
88150-59-8
|
98%
|
|
UK51656 is an antagonist of calcium (IC50: 4 nM).
|
T15553 |
Iganidipine
|
119687-33-1
|
98%
|
|
Iganidipine is an antagonist of Ca2+ .
|
T13117 |
Teludipine hydrochloride
|
108700-03-4
|
98%
|
|
Teludipine hydrochloride is a blocker of lipophilic calcium channel.
|
TN3660 |
Cinnamyl caffeate
|
115610-32-7
|
98%
|
|
Cinnamyl caffeate has cardiovascular protective effects, it can increase H9c2 cellular antioxidant potential, decrease intracellular calcium ion ([Ca2+]i) level,...
|
TN1588 |
Dihydroisotanshinone I
|
20958-18-3
|
98%
|
|
Dihydroisotanshinone I has protective action against menadione-induced hepatotoxicity, attributed to its antioxidant properties including the free radical scaven...
|
TP1852 |
Myomodulin
|
110570-93-9
|
98%
|
|
Myomodulin is a neuropeptide present in molluscs, insects, and gastropods.Myomodulin is present in two identified aplysia neurons that contain myomodulin A the A...
|
T19253 |
Cyclic ADP-ribose
|
119340-53-3
|
98%
|
|
Cyclic ADP-ribose (cADPR) is an effective calcium mobilization second messenger, which is synthesized from NAD + by ADP-ribosyl cyclase. Cyclic ADP-ribose mainly...
|
TN2211 |
Silybin B
|
142797-34-0
|
98%
|
|
Silybin B and silybin A are potent inhibitors of both raloxifene 4'- and 6-glucuronidation in all enzyme systems; they show strong effects on cell growth inhibit...
|
TMA0805 |
Lupanine
|
550-90-3
|
98%
|
|
Lupanine has a weak sedative effect on the central nervous system, interaction with specific drugs used for treatment of the CNS and for analgesic activity. Lupa...
|