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Calcium Channel

A calcium channel is an ion channel which shows selective permeability to calcium ions. It is sometimes synonymous with voltage-gated calcium channel, although there are also ligand-gated calcium channels.
Cat No. product name
T9888 YM-244769 YM-244769 是一种有效的 Na+/Ca2+ exchange 3 (NCX3) 抑制剂,IC50 为 18 nM。 YM-244769 对神经元和肾脏具有有效的保护作用。
T39195 YM-244769 dihydrochloride YM-244769 dihydrochloride 是一种有效的 Na+/Ca2+ exchange 3 (NCX3) 抑制剂,IC50 为 18 nM。 YM-244769 dihydrochloride 对神经元和肾脏具有有效的保护作用。
T15366 Gabapentin enacarbil Gabapentin enacarbil 是抗惊厥和镇痛药物加巴喷丁的前药。Gabapentin enacarbil 提供持续剂量比例的 Gabapentin 暴露和可预测的生物利用度。
T24984 5J-4 5J-4 是一种有效的钙释放激活钙通道 (CRAC) 和钙池操纵性钙内流(SOCE) 阻滞剂。 5J-4 减少 IL-17 的产生并降低 RORα 和 RORγt 的表达。
T4S1419 (±)-Praeruptorin A 1. Praeruptorin A could exhibit its anti-osteoclastogenic activity by inhibiting p38/Akt-c-Fos-NFATc1 signaling and PLCγ-independent Ca(2+) oscillation 2. Praeru...
T7540 2,5-Di-tert-butylhydroquinone BHQ is an effective and selective endoplasmic reticulum Ca2+-ATPase inhibitor.
T3524 Halofuginone hydrobromide Halofuginone specifically inhibits collagen type I gene expression and matrix metalloproteinase 2 (MMP-2) gene expression, which may result in the suppression of...
T1435 Praziquantel Praziquantel increases the permeability of the tegument of susceptible worms, resulting in an influx and increase in intra-tegumental calcium leading to rapid co...
T15053 Darodipine Darodipine is a potent antagonist of calcium channel.
TP1852 Myomodulin Myomodulin is a neuropeptide present in molluscs, insects, and gastropods.Myomodulin is present in two identified aplysia neurons that contain myomodulin A the A...
T6856 Halofuginone Halofuginone, the competitive inhibitor of prolyl-tRNA synthetase(Ki=18.3 nM), could also down-regulate Smad3 and blocked TGF-β signaling at 10 ng/ml in the mamm...
T10885 CRAC intermediate 2 CRAC intermediate 2 is a intermediate compound for CRAC inhibitor synthesis. CRAC intermediate 2 has been extracted from patent WO 2013059666A1.
T4054 Dantrolene sodium hemiheptahydrate Dantrolene depresses excitation-contraction coupling in skeletal muscle by binding to the ryanodine receptor 1 and decreasing intracellular calcium concentration...
T0858 Flufenamic acid Flufenamic acid is an anthranilic acid derivative with analgesic, anti-inflammatory, and antipyretic properties. It is used in musculoskeletal and joint disorder...
TN1757 Hypophyllanthin Hypophyllanthin and phyllanthin have antitumour effects against Ehrlich Ascites Carcinoma in mice.
T5701 OPHIOPOGONIN D Ophiopogonin D is a natural product,and is a CYP2J3 inducer that significantly inhibits Ang II induced NF-κB nuclear translocation.
T6227 Benidipine hydrochloride Benidipine HCl, a hydrochloride salt form of benidipine, is used as a blocker of dihydropyridine calcium channel.
T1198 Tetracaine hydrochloride Tetracaine hydrochloride (Pontocaine), a potent local anaesthetic, is a channel function allosteric inhibitor. It is primarily used as an antipruritic and topica...
T29201 Z944 Z944 is an antagonist of T-type calcium channel. Z944 Delays the Progression of Seizures in the Amygdala Kindling Model. Z944 disrupts prepulse inhibition in bot...
T2782 Catharanthine Catharanthine suppresses nicotinic receptor-mediated diaphragm contractions (IC50=59.6 μM).
T6S1418 Praeruptorin C 1. Praeruptorin C has been widely used as an antioxidant and a calcium antagonist to treat diseases. 2. Praeruptorin C partially protects cortical neurons by inh...
T1439 Lacidipine Lacidipine is a lipophilic dihydropyridine calcium antagonist with an intrinsically slow onset of activity. Due to its long duration of action, lacidipine does n...
T1073 Dronedarone hydrochloride Dronedarone hydrochloride is an amiodarone analog which has an effective and promising treatment for Atrial fibrillation.
TN7108 Urolithin C Urolithin C is a gut metabolite of ellagic acid. Urolithin C induces apoptosis in PC12 cells through a mitochondria-mediated pathway.
TN1008 Psoralenoside Psoralenoside is a natural product isolated from the fruits of Psoralea corylifolia, shows estrogen-like activity, osteoblastic proliferation accelerating activi...
T0825 Ebselen Ebselen is a organoselenium compound with anti-inflammatory, anti-oxidant and cytoprotective activity. Ebselen acts as a glutathione peroxidase mimetic and is th...
T1730 NPS-2143 NPS-2143 is a novel potent and selective antagonist of Ca(2+) receptor.
T10024 1-Octanol 1-Octanol (Octanol), a saturated fatty alcohol, is a T-type calcium channels (T-channels) inhibitor with an IC50 of 4 μM for native T-currents[1]. 1-Octanol is a...
TN5073 Strophanthidin Strophanthidin can induce calcium overload in vivo.
TN1721 Gypenoside L Gypenoside L inhibits autophagic flux and induces cell death in human esophageal cancer cells through endoplasm reticulum stress-mediated Ca2+ release. It also i...
T5114 Pyridaben Pyridaben is a METI acaricide that inhibits mitochondrial electron transport at complex I (METI; Ki = 0.36 nmol/mg protein in rat brain mitochondria).
T0928 L-Ascorbic acid Vitamin C is a potent reducing and antioxidant agent that functions in fighting bacterial infections, in detoxifying reactions, and in the formation of collagen....
T1105 Penfluridol Penfluridol is a highly potent antipsychotic.
T11665 Ionomycin calcium lonomycin calcium is a potent, selective calcium ionophore and an antibiotic produced by Streptomyces conglobatus. also induces the activation of protein kinase ...
T3013 Catharanthine tartrate Extracted from whole herb of Catharanthus roseus (L.)G.Don;Store the product in sealed, cool and dry condition.
T0916 Butamben Butamben is a long-duration local anesthetic used for the treatment of chronic pain.
T0192 Levetiracetam Levetiracetam is a relatively unique anticonvulsant that is typically used in combination with other antiepileptic medications for partial onset seizures. Leveti...
T1215 Nicardipine hydrochloride Nicardipine Hydrochloride is the hydrochloride salt form of nicardipine, a synthetic derivative of nitrophenyl-pyridine and potent calcium channel blocker, Nicar...
T0163 Nisoldipine Nisoldipine is a dihydropyridine calcium channel antagonist that acts as a potent arterial vasodilator and antihypertensive agent.
T1260 Cromolyn sodium Cromolyn sodium is a chromone complex that acts by inhibiting the release of chemical mediators from sensitized mast cells.
T4669 Fantofarone Fantofarone is a highly potent Calcium Channel antagonist.
T6S0659 Rhynchophylline 1. Rhynchophylline can protect against ischemic damage, probably via regulating the Akt/mTOR pathway. 2. Rhynchophylline can protect against glutamate-induced ne...
T0207 Ranolazine dihydrochloride Ranolazine(RS-43285), an antianginal agent, can treat arrhythmia via a novel mechanism of action (inhibition of the late phase of the inward sodium current), and...
T2170 SKF-96365 hydrochloride SKF-96365, a SOCE inhibitor, exhibits potent anti-neoplastic activity by inducing cell-cycle arrest and apoptosis in colorectal Y cells. SKF-96365 can induce cyt...
T13047 Synta66 Synta66 is a store-operated calcium entry channel Orai inhibitor, and used for the research of neurological disease.
T2003 ISX-9 ISX9 is necessary to activate neuron-specific genes as neurogenesis inducer.
T1010 Verapamil hydrochloride Verapamil hydrochloride is a calcium channel blocker that is a class IV anti-arrhythmia agent.
T0145 Felodipine Felodipine is a longlasting 1, 4-dihydropyridine calcium channel repressor.
TN1624 Ethyl cinnamate Ethyl cinnamate has antifungal, and vasorelaxant effects, it can inhibit the tonic contractions induced by high K+ and phenylephrine (PE) in a concentration-depe...
T22353 Lanthanum(III) chloride heptahydrate Lanthanum(III) chloride is an inorganic compound which used in biochemical research to block the activity of divalent cation channels, especially calcium channel...
YM-244769
T9888
YM-244769 是一种有效的 Na+/Ca2+ exchange 3 (NCX3) 抑制剂,IC50 为 18 nM。 YM-244769 对神经元和肾脏具有有效的保护作用。
YM-244769 dihydrochloride
T39195
YM-244769 dihydrochloride 是一种有效的 Na+/Ca2+ exchange 3 (NCX3) 抑制剂,IC50 为 18 nM。 YM-244769 dihydrochloride 对神经元和肾脏具有有效...
Gabapentin enacarbil
T15366
5J-4
T24984
(±)-Praeruptorin A
T4S1419
1. Praeruptorin A could exhibit its anti-osteoclastogenic activity by inhibiting p38/Akt-c-Fos-NFATc1 signaling and PLCγ-independent Ca(2+) oscillation 2. Praer...
2,5-Di-tert-butylhydroquinone
T7540
BHQ is an effective and selective endoplasmic reticulum Ca2+-ATPase inhibitor.
Halofuginone hydrobromide
T3524
Halofuginone specifically inhibits collagen type I gene expression and matrix metalloproteinase 2 (MMP-2) gene expression, which may result in the suppression of...
Praziquantel
T1435
Praziquantel increases the permeability of the tegument of susceptible worms, resulting in an influx and increase in intra-tegumental calcium leading to rapid co...
Darodipine
T15053
Darodipine is a potent antagonist of calcium channel.
Myomodulin
TP1852
Myomodulin is a neuropeptide present in molluscs, insects, and gastropods.Myomodulin is present in two identified aplysia neurons that contain myomodulin A the A...
Halofuginone
T6856
Halofuginone, the competitive inhibitor of prolyl-tRNA synthetase(Ki=18.3 nM), could also down-regulate Smad3 and blocked TGF-β signaling at 10 ng/ml in the...
CRAC intermediate 2
T10885
CRAC intermediate 2 is a intermediate compound for CRAC inhibitor synthesis. CRAC intermediate 2 has been extracted from patent WO 2013059666A1.
Dantrolene sodium hemiheptahydrate
T4054
Dantrolene depresses excitation-contraction coupling in skeletal muscle by binding to the ryanodine receptor 1 and decreasing intracellular calcium concentration...
Flufenamic acid
T0858
Flufenamic acid is an anthranilic acid derivative with analgesic, anti-inflammatory, and antipyretic properties. It is used in musculoskeletal and joint disorder...
Hypophyllanthin
TN1757
Hypophyllanthin and phyllanthin have antitumour effects against Ehrlich Ascites Carcinoma in mice.
OPHIOPOGONIN D
T5701
Ophiopogonin D is a natural product,and is a CYP2J3 inducer that significantly inhibits Ang II induced NF-κB nuclear translocation.
Benidipine hydrochloride
T6227
Benidipine HCl, a hydrochloride salt form of benidipine, is used as a blocker of dihydropyridine calcium channel.
Tetracaine hydrochloride
T1198
Tetracaine hydrochloride (Pontocaine), a potent local anaesthetic, is a channel function allosteric inhibitor. It is primarily used as an antipruritic and topica...
Z944
T29201
Z944 is an antagonist of T-type calcium channel. Z944 Delays the Progression of Seizures in the Amygdala Kindling Model. Z944 disrupts prepulse inhibition in bot...
Catharanthine
T2782
Catharanthine suppresses nicotinic receptor-mediated diaphragm contractions (IC50=59.6 μM).
Praeruptorin C
T6S1418
1. Praeruptorin C has been widely used as an antioxidant and a calcium antagonist to treat diseases. 2. Praeruptorin C partially protects cortical neurons by inh...
Lacidipine
T1439
Lacidipine is a lipophilic dihydropyridine calcium antagonist with an intrinsically slow onset of activity. Due to its long duration of action, lacidipine does n...
Dronedarone hydrochloride
T1073
Dronedarone hydrochloride is an amiodarone analog which has an effective and promising treatment for Atrial fibrillation.
Urolithin C
TN7108
Urolithin C is a gut metabolite of ellagic acid. Urolithin C induces apoptosis in PC12 cells through a mitochondria-mediated pathway.
Psoralenoside
TN1008
Psoralenoside is a natural product isolated from the fruits of Psoralea corylifolia, shows estrogen-like activity, osteoblastic proliferation accelerating activi...
Ebselen
T0825
Ebselen is a organoselenium compound with anti-inflammatory, anti-oxidant and cytoprotective activity. Ebselen acts as a glutathione peroxidase mimetic and is th...
NPS-2143
T1730
NPS-2143 is a novel potent and selective antagonist of Ca(2+) receptor.
1-Octanol
T10024
1-Octanol (Octanol), a saturated fatty alcohol, is a T-type calcium channels (T-channels) inhibitor with an IC50 of 4 μM for native T-currents[1]. 1-Octanol is ...
Strophanthidin
TN5073
Strophanthidin can induce calcium overload in vivo.
Gypenoside L
TN1721
Gypenoside L inhibits autophagic flux and induces cell death in human esophageal cancer cells through endoplasm reticulum stress-mediated Ca2+ release. It also i...
Pyridaben
T5114
Pyridaben is a METI acaricide that inhibits mitochondrial electron transport at complex I (METI; Ki = 0.36 nmol/mg protein in rat brain mitochondria).
L-Ascorbic acid
T0928
Vitamin C is a potent reducing and antioxidant agent that functions in fighting bacterial infections, in detoxifying reactions, and in the formation of collagen....
Penfluridol
T1105
Penfluridol is a highly potent antipsychotic.
Ionomycin calcium
T11665
lonomycin calcium is a potent, selective calcium ionophore and an antibiotic produced by Streptomyces conglobatus. also induces the activation of protein kinase ...
Catharanthine tartrate
T3013
Extracted from whole herb of Catharanthus roseus (L.)G.Don;Store the product in sealed, cool and dry condition.
Butamben
T0916
Butamben is a long-duration local anesthetic used for the treatment of chronic pain.
Levetiracetam
T0192
Levetiracetam is a relatively unique anticonvulsant that is typically used in combination with other antiepileptic medications for partial onset seizures. Leveti...
Nicardipine hydrochloride
T1215
Nicardipine Hydrochloride is the hydrochloride salt form of nicardipine, a synthetic derivative of nitrophenyl-pyridine and potent calcium channel blocker, Nicar...
Nisoldipine
T0163
Nisoldipine is a dihydropyridine calcium channel antagonist that acts as a potent arterial vasodilator and antihypertensive agent.
Cromolyn sodium
T1260
Cromolyn sodium is a chromone complex that acts by inhibiting the release of chemical mediators from sensitized mast cells.
Fantofarone
T4669
Fantofarone is a highly potent Calcium Channel antagonist.
Rhynchophylline
T6S0659
1. Rhynchophylline can protect against ischemic damage, probably via regulating the Akt/mTOR pathway. 2. Rhynchophylline can protect against glutamate-induced ne...
Ranolazine dihydrochloride
T0207
Ranolazine(RS-43285), an antianginal agent, can treat arrhythmia via a novel mechanism of action (inhibition of the late phase of the inward sodium current), and...
SKF-96365 hydrochloride
T2170
SKF-96365, a SOCE inhibitor, exhibits potent anti-neoplastic activity by inducing cell-cycle arrest and apoptosis in colorectal Y cells. SKF-96365 can induce cyt...
Synta66
T13047
Synta66 is a store-operated calcium entry channel Orai inhibitor, and used for the research of neurological disease.
ISX-9
T2003
ISX9 is necessary to activate neuron-specific genes as neurogenesis inducer.
Verapamil hydrochloride
T1010
Verapamil hydrochloride is a calcium channel blocker that is a class IV anti-arrhythmia agent.
Felodipine
T0145
Felodipine is a longlasting 1, 4-dihydropyridine calcium channel repressor.
Ethyl cinnamate
TN1624
Ethyl cinnamate has antifungal, and vasorelaxant effects, it can inhibit the tonic contractions induced by high K+ and phenylephrine (PE) in a concentration-depe...
Lanthanum(III) chloride heptahydrate
T22353
Lanthanum(III) chloride is an inorganic compound which used in biochemical research to block the activity of divalent cation channels, especially calcium channel...
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