Adrenergic Receptor

The adrenergic receptors or adrenoceptors are a class of G protein-coupled receptors that are targets of many catecholamines like norepinephrine (noradrenaline) and epinephrine (adrenaline) produced by the body, but also many medications like beta blockers, β2 agonists and α2 agonists, which are used to treat high blood pressure and asthma, for example.

Cat. No.	Product name	CAS No.	Purity
TN4882	Quinine HCl	130-89-2	98%
TN4882	Quinine HCl produces alpha-adrenergic blockade. Quinine modifies catecholamine- and calcium-induced myocardial contractile force responses.
T11036	Diacetolol D7	1346604-19-0	98%
T11036	Diacetolol D7 is deuterium-labeled diacetone Roller. Diacetol is the main metabolite of Acetolol. Diacetololβ-adrenoceptor shielding and anti-arrhythmic agent.
T23557	Talibegron hydrochloride	178600-17-4	98%
T23557	Talibegron hydrochloride is an β3 adrenergic receptor agonist with a pD2 of 3.72 on phenylephrine-preconstricted rat mesenteric artery. Relaxes rat mesenteric ar...
T6860	ICI-118551 Hydrochloride	1217094-53-5	98%
T6860	ICI-118551 is a highly selective β2-adrenergic receptor antagonist with Ki values of 0.7, 49.5 and 611 nM for β2, β1 and β3 receptors, respectively.
T12815	(S)-Terazosin	109351-33-9	98%
T12815	(S)-Terazosin is an active S-enantiomer of Terazosin. (S)-Terazosin is a potent and high-affinity antagonist of α-adrenoceptor(α1a, α1b and α1d-adrenoceptor with...
T13470	(±)-Levomepromazine-d6	1189805-51-3	98%
T13470	(±)-Methotrimeprazine (D6) is the deuterium labeled Methotrimeprazine, which is an antagonist of D3 dopamine and Histamine H1 receptor.
T10778	CGP 20712 A	105737-62-0	98%
T10778	CGP 20712 A (CGP 20712 mesylate) is a highly selective antagonist of β1-adrenoceptor (IC50: 0.7 nM). It shows ~10,000-fold selectivity over β2-adrenoceptors.
TCS2185	Yohimbine	146-48-5	98%
TCS2185	Yohimbine is a nonselective alpha 2-adrenergic receptor (AR) antagonist(IC50 : 0.6 μM)
T1728	Lofexidine hydrochloride	21498-08-8	98%
T1728	Lofexidine (hydrochloride) is a selective α2-receptor agonist, commonly used to alleviate the physical symptoms of heroin and other types of opioid withdrawal [1...
T13403	ZK-90055 hydrochloride	84638-81-3	98%
T13403	ZK-90055 hydrochloride is an agonist of β2 adrenergic receptor.
T6663	Scopine hydrochloride	85700-55-6	98%
T6663	Scopine HCl salt is the metabolite of anisodine, which is a α1-adrenergic receptor agonist and used in the treatment of acute circulatory shock.
T10364	Arbutamine	128470-16-6	98%
T10364	Arbutamine is a short-acting synthetic potent nonselective β-adrenoceptor agonist that increases cardiac contractility, heart rate, and systolic blood pressure.
TN5061	Stephanine	517-63-5	98%
TN5061	l-Stephanine is a potent and highly selective alpha 1 adrenoceptor blocker, inhibits anococcygeus muscle contraction induced by phenylephrine with pA2 values of ...
T7065	Tizanidine	51322-75-9	98%
T7065	Tizanidine is an α2-adrenergic receptor agonist and inhibits neurotransmitter release from CNS noradrenergic neurons.
T5450	DL-071-IT	55104-39-7	98%
T5450	DL 071-IT is a potent non-selective beta-adrenoceptor antagonist. DL 071 IT showed intrinsic sympathomimetic activity and weak membrane stabilizing activity.
T13285	Vatinoxan hydrochloride	130466-38-5	98%
T13285	Vatinoxan hydrochloride is an antagonist of the peripheral α2 adrenergic receptors.
T14287	Ancarolol	75748-50-4	98%
T14287	Ancarolol is a blocking agent of beta-adrenergic.
T13804	OPC-28326	167626-17-7	98%
T13804	OPC-28326 is a specific an α2-adrenergic receptor antagonist and acts as a peripheral vasodilator. OPC-28326 inhibits α2A-, α2B- and α2C-adrenoceptors with Ki of...
T6562	Latrepirdine dihydrochloride	97657-92-6	98%
T6562	Latrepirdine is an orally active, and neuroactive antagonist of multiple drug targets, including histamine receptors, GluR, and 5-HT receptors, used as an antihi...
T11015	Midaglizole hydrochloride	79689-25-1	98%
T11015	Midaglizole hydrochloride (DG5128) is a preferred α2-adrenoceptor antagonist. Midazolazole hydrochloride (DG5128) has an affinity for α2-adrenoceptor (pKi = 6.28...