TN4882 |
Quinine HCl
|
130-89-2
|
98%
|
|
Quinine HCl produces alpha-adrenergic blockade. Quinine modifies catecholamine- and calcium-induced myocardial contractile force responses.
|
T11036 |
Diacetolol D7
|
1346604-19-0
|
98%
|
|
Diacetolol D7 is deuterium-labeled diacetone Roller. Diacetol is the main metabolite of Acetolol. Diacetololβ-adrenoceptor shielding and anti-arrhythmic agent.
|
T23557 |
Talibegron hydrochloride
|
178600-17-4
|
98%
|
|
Talibegron hydrochloride is an β3 adrenergic receptor agonist with a pD2 of 3.72 on phenylephrine-preconstricted rat mesenteric artery. Relaxes rat mesenteric ar...
|
T6860 |
ICI-118551 Hydrochloride
|
1217094-53-5
|
98%
|
|
ICI-118551 is a highly selective β2-adrenergic receptor antagonist with Ki values of 0.7, 49.5 and 611 nM for β2, β1 and β3 receptors, respectively.
|
T12815 |
(S)-Terazosin
|
109351-33-9
|
98%
|
|
(S)-Terazosin is an active S-enantiomer of Terazosin. (S)-Terazosin is a potent and high-affinity antagonist of α-adrenoceptor(α1a, α1b and α1d-adrenoceptor with...
|
T13470 |
(±)-Levomepromazine-d6
|
1189805-51-3
|
98%
|
|
(±)-Methotrimeprazine (D6) is the deuterium labeled Methotrimeprazine, which is an antagonist of D3 dopamine and Histamine H1 receptor.
|
T10778 |
CGP 20712 A
|
105737-62-0
|
98%
|
|
CGP 20712 A (CGP 20712 mesylate) is a highly selective antagonist of β1-adrenoceptor (IC50: 0.7 nM). It shows ~10,000-fold selectivity over β2-adrenoceptors.
|
TCS2185 |
Yohimbine
|
146-48-5
|
98%
|
|
Yohimbine is a nonselective alpha 2-adrenergic receptor (AR) antagonist(IC50 : 0.6 μM)
|
T1728 |
Lofexidine hydrochloride
|
21498-08-8
|
98%
|
|
Lofexidine (hydrochloride) is a selective α2-receptor agonist, commonly used to alleviate the physical symptoms of heroin and other types of opioid withdrawal [1...
|
T13403 |
ZK-90055 hydrochloride
|
84638-81-3
|
98%
|
|
ZK-90055 hydrochloride is an agonist of β2 adrenergic receptor.
|
T6663 |
Scopine hydrochloride
|
85700-55-6
|
98%
|
|
Scopine HCl salt is the metabolite of anisodine, which is a α1-adrenergic receptor agonist and used in the treatment of acute circulatory shock.
|
T10364 |
Arbutamine
|
128470-16-6
|
98%
|
|
Arbutamine is a short-acting synthetic potent nonselective β-adrenoceptor agonist that increases cardiac contractility, heart rate, and systolic blood pressure.
|
TN5061 |
Stephanine
|
517-63-5
|
98%
|
|
l-Stephanine is a potent and highly selective alpha 1 adrenoceptor blocker, inhibits anococcygeus muscle contraction induced by phenylephrine with pA2 values of ...
|
T7065 |
Tizanidine
|
51322-75-9
|
98%
|
|
Tizanidine is an α2-adrenergic receptor agonist and inhibits neurotransmitter release from CNS noradrenergic neurons.
|
T5450 |
DL-071-IT
|
55104-39-7
|
98%
|
|
DL 071-IT is a potent non-selective beta-adrenoceptor antagonist. DL 071 IT showed intrinsic sympathomimetic activity and weak membrane stabilizing activity.
|
T13285 |
Vatinoxan hydrochloride
|
130466-38-5
|
98%
|
|
Vatinoxan hydrochloride is an antagonist of the peripheral α2 adrenergic receptors.
|
T14287 |
Ancarolol
|
75748-50-4
|
98%
|
|
Ancarolol is a blocking agent of beta-adrenergic.
|
T13804 |
OPC-28326
|
167626-17-7
|
98%
|
|
OPC-28326 is a specific an α2-adrenergic receptor antagonist and acts as a peripheral vasodilator. OPC-28326 inhibits α2A-, α2B- and α2C-adrenoceptors with Ki of...
|
T6562 |
Latrepirdine dihydrochloride
|
97657-92-6
|
98%
|
|
Latrepirdine is an orally active, and neuroactive antagonist of multiple drug targets, including histamine receptors, GluR, and 5-HT receptors, used as an antihi...
|
T11015 |
Midaglizole hydrochloride
|
79689-25-1
|
98%
|
|
Midaglizole hydrochloride (DG5128) is a preferred α2-adrenoceptor antagonist. Midazolazole hydrochloride (DG5128) has an affinity for α2-adrenoceptor (pKi = 6.28...
|