Dopamine Receptor

Dopamine receptors are a class of G protein-coupled receptors that are prominent in the vertebrate central nervous system (CNS). Dopamine receptors activate different effectors through not only G-protein coupling, but also signaling through different protein (dopamine receptor-interacting proteins) interactions.

Cat. No.	Product name	CAS No.	Purity
T13652	Dicarbine	17411-19-7	98%
T13652	Double carbene can be used for the study of schizophrenia and alcoholism. It can block dopamine receptors in various parts of the brain and prevent the reduction...
T16511	PF2562	1609258-91-4	98%
T16511	PF2562 is a dopamine D1 ligand. It is used as a dopamine D1 agonist or partial agonist. PF2562 binds to human D1 receptor (Ki: 113 nM). PF2562 shows activity aga...
T12676	(Rac)-Rotigotine hydrochloride	102120-99-0	98%
T12676	(Rac)-Rotigotine hydrochloride is a racemate of Rotigotine. Rotigotine is a full agonist of dopamine receptor, a partial the 5-HT1A receptor agonist.
T12861L	SB-277011 dihydrochloride	1226917-67-4	98%
T12861L	SB-277011 dihydrochloride is a potent, selective, orally bioavailable and brain penetrate antagonist of dopamine D3 receptor(pKis of 8.0, 6.0, <5.2 and 5.9 for D...
T12288	Odapipam	131796-63-9	98%
T12288	Odapipam is a selective and high affinity antagonist of benzazepine dopamine D1 receptor (Kd of 0.18 nM).
T1769	Pardoprunox	269718-84-5	98%
T1769	Pardoprunox is a partial dopamine D2 agonist and noradrenergic agonist with serotonin 5-HT1A agonist properties. Pardoprunox has been used in trials studying the...
T3086	Mesoridazine Besylate	32672-69-8	98%
T3086	Mesoridazine (Serentil) is a piperidine neuroleptic drug belonging to the class of drugs called phenothiazines, used in the treatment of schizophrenia. It is a m...
T13240	U91356	152886-85-6	98%
T13240	U91356 is an agonist of the dopamine receptors.
T11799L	L-745870	158985-00-3	98%
T11799L	L-745870 is a high-affinity and selective human dopamine D4 receptor antagonist (Ki: 0.43 nM). L-745870 has excellent brain penetration. It considerably weaker D...
T67729	UCM-1306	2258608-78-3	98%
T67729	UCM-1306 is a potent and orally active allosteric modulator (PAM) of human dopamine D1 receptor. UCM-1306 could increase the maximal effect of endogenous dopamin...
T15744	Levophacetoperane hydrochloride	23257-56-9	98%
T15744	Levophacetoperane inhibits in vitro in a competitive manner. It also can norepinephrine uptake and dopamine uptake.
T7341	Diclofensine	67165-56-4	98%
T7341	Diclofensine inhibits the uptake of serotonin, noradrenaline and dopamine.
T15117	Didesmethyl cariprazine	839712-25-3	98%
T15117	Cariprazine is an antipsychotic drug candidate. It shows high affinity for the D3 and D2 receptors, and moderate affinity for the 5-HT1A receptor. Didesmethyl ca...
T10213	A-437203	220519-06-2	98%
T10213	A-437203 is a selective D3 receptor antagonist (Kis: 71, 1.6, and 6220 nM for D2, D3, and D4 receptors).
TQ0140	Sumanirole maleate	179386-44-8	98%
TQ0140	Sumanirole maleate (U-95666E) is a highly selective full agonist of the D2 receptor (ED50: 46 nM).
T6142	PD128907 HCl	112960-16-4	98%
T6142	PD128907 HCl 是一种有效的选择性多巴胺 D3 受体激动剂，EC50 为 0.64 nM，选择性是多巴胺 D2 受体的 53 倍。
T4007	Eticlopride hydrochloride	97612-24-3	98%
T4007	Eticlopride, an antipsychotic, is a Selective dopamine D2/D3 receptor antagonist (Ki: 0.5/0.16 nM).
T2S1397	L-Stepholidine	16562-13-3	98%
T2S1397	L-Stepholidine, which has dual actions on dopamine D1 and D2 receptors, attenuates heroin self-administration and cue-induced reinstatement. It also elicits anti...
T15339	Foscarbidopa	1907685-81-7	98%
T15339	Foscarbidopa is a prodrug of Carbidopa. It acts as a dopamine receptor agonist.
T9237	Rotigotine	92206-54-7	98%
T9237	Rotigotine is an antiparkinson agent and dopamine receptor agonist.