T13652 |
Dicarbine
|
17411-19-7
|
98%
|
|
Double carbene can be used for the study of schizophrenia and alcoholism. It can block dopamine receptors in various parts of the brain and prevent the reduction...
|
T16511 |
PF2562
|
1609258-91-4
|
98%
|
|
PF2562 is a dopamine D1 ligand. It is used as a dopamine D1 agonist or partial agonist. PF2562 binds to human D1 receptor (Ki: 113 nM). PF2562 shows activity aga...
|
T12676 |
(Rac)-Rotigotine hydrochloride
|
102120-99-0
|
98%
|
|
(Rac)-Rotigotine hydrochloride is a racemate of Rotigotine. Rotigotine is a full agonist of dopamine receptor, a partial the 5-HT1A receptor agonist.
|
T12861L |
SB-277011 dihydrochloride
|
1226917-67-4
|
98%
|
|
SB-277011 dihydrochloride is a potent, selective, orally bioavailable and brain penetrate antagonist of dopamine D3 receptor(pKis of 8.0, 6.0, <5.2 and 5.9 for D...
|
T12288 |
Odapipam
|
131796-63-9
|
98%
|
|
Odapipam is a selective and high affinity antagonist of benzazepine dopamine D1 receptor (Kd of 0.18 nM).
|
T1769 |
Pardoprunox
|
269718-84-5
|
98%
|
|
Pardoprunox is a partial dopamine D2 agonist and noradrenergic agonist with serotonin 5-HT1A agonist properties. Pardoprunox has been used in trials studying the...
|
T3086 |
Mesoridazine Besylate
|
32672-69-8
|
98%
|
|
Mesoridazine (Serentil) is a piperidine neuroleptic drug belonging to the class of drugs called phenothiazines, used in the treatment of schizophrenia. It is a m...
|
T13240 |
U91356
|
152886-85-6
|
98%
|
|
U91356 is an agonist of the dopamine receptors.
|
T11799L |
L-745870
|
158985-00-3
|
98%
|
|
L-745870 is a high-affinity and selective human dopamine D4 receptor antagonist (Ki: 0.43 nM). L-745870 has excellent brain penetration. It considerably weaker D...
|
T67729 |
UCM-1306
|
2258608-78-3
|
98%
|
|
UCM-1306 is a potent and orally active allosteric modulator (PAM) of human dopamine D1 receptor. UCM-1306 could increase the maximal effect of endogenous dopamin...
|
T15744 |
Levophacetoperane hydrochloride
|
23257-56-9
|
98%
|
|
Levophacetoperane inhibits in vitro in a competitive manner. It also can norepinephrine uptake and dopamine uptake.
|
T7341 |
Diclofensine
|
67165-56-4
|
98%
|
|
Diclofensine inhibits the uptake of serotonin, noradrenaline and dopamine.
|
T15117 |
Didesmethyl cariprazine
|
839712-25-3
|
98%
|
|
Cariprazine is an antipsychotic drug candidate. It shows high affinity for the D3 and D2 receptors, and moderate affinity for the 5-HT1A receptor. Didesmethyl ca...
|
T10213 |
A-437203
|
220519-06-2
|
98%
|
|
A-437203 is a selective D3 receptor antagonist (Kis: 71, 1.6, and 6220 nM for D2, D3, and D4 receptors).
|
TQ0140 |
Sumanirole maleate
|
179386-44-8
|
98%
|
|
Sumanirole maleate (U-95666E) is a highly selective full agonist of the D2 receptor (ED50: 46 nM).
|
T6142 |
PD128907 HCl
|
112960-16-4
|
98%
|
|
PD128907 HCl 是一种有效的选择性多巴胺 D3 受体激动剂,EC50 为 0.64 nM,选择性是多巴胺 D2 受体的 53 倍。
|
T4007 |
Eticlopride hydrochloride
|
97612-24-3
|
98%
|
|
Eticlopride, an antipsychotic, is a Selective dopamine D2/D3 receptor antagonist (Ki: 0.5/0.16 nM).
|
T2S1397 |
L-Stepholidine
|
16562-13-3
|
98%
|
|
L-Stepholidine, which has dual actions on dopamine D1 and D2 receptors, attenuates heroin self-administration and cue-induced reinstatement. It also elicits anti...
|
T15339 |
Foscarbidopa
|
1907685-81-7
|
98%
|
|
Foscarbidopa is a prodrug of Carbidopa. It acts as a dopamine receptor agonist.
|
T9237 |
Rotigotine
|
92206-54-7
|
98%
|
|
Rotigotine is an antiparkinson agent and dopamine receptor agonist.
|