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Dopamine Receptor

Dopamine receptors are a class of G protein-coupled receptors that are prominent in the vertebrate central nervous system (CNS). Dopamine receptors activate different effectors through not only G-protein coupling, but also signaling through different protein (dopamine receptor-interacting proteins) interactions.
Cat No. product name
T22019 ABT 724 trihydrochloride ABT 724 trihydrochloride 是一种有效的选择性 D4 受体激动剂(EC50 = 12.4 nM,14.3 nM 和 23.2 nM,分别对人、大鼠和雪貂)。 ABT-724 trihydrochloride 可用于勃起功能障碍研究。
T1644 Dopamine hydrochloride Dopamine is a naturally occurring catecholamine formed by decarboxylation of dihydroxyphenylalanine and a precursor of norepinephrine and epinephrine. Dopamine b...
T1540 Doxepin hydrochloride Doxepin Hydrochloride is a dibenzoxepin tricyclic compound. It displays a range of pharmacological actions including maintaining adrenergic innervation. Its mech...
T0505 Methyldopa Methyldopa, an alpha-adrenergic agonist (selective for α2-adrenergic receptors) psychoactive medicine, is served as an antihypertensive or sympatholytic.
T24047 Etilevodopa hydrochloride Etilevodopa HCl is a prodrug of levodopa. It also has greater gastric solubility and significant brain penetration.
T0848 L-DOPA Levodopa is an amino acid precursor of dopamine with antiparkinsonian properties. Levodopa is a prodrug that is converted to dopamine by DOPA decarboxylase and c...
T0074 Chlorprothixene Chlorprothixene is a typical antipsychotic drug of the thioxanthene class, which was the first of the series to be synthesized.
T2631 WAY-100635 Maleate WAY-100635 is a specific and effective 5-HT receptor antagonist (IC50=0.95 nM).
T8385 Metoclopramide hydrochloride hydrate Metoclopramide hydrochloride hydrate is a dopamine D2 antagonist that is a drug used for digestive dysfunction. It acts as an anti-emetic
T22508 3-CPMT dopamine uptake inhibitor
T12865 SCH-23390 maleate SCH-23390 maleate is a potent and selective antagonist of dopamine D1-like receptor (1 and D5 receptor with Kis of 0.2 nM and 0.3 nM, respectively).
T35841 5-Benzyloxygramine 5-Benzyloxygramine is a N protein PPI orthosteric stabilizer that exhibits both antiviral and N-NTD protein-stabilizing activities[1]. 5-benzyloxygramine stabili...
T1539 Iloperidone Iloperidone is an atypical antipsychotic agent that is used for treatment of schizophrenia.
T2917 Tetrahydropalmatine hydrochloride Tetrahydropalmatine (THP) is an isoquinoline alkaloid found in several different plant species, mainly in the Corydalis genus (Yan Hu Suo). It is a potent muscle...
T4616 Metoclopramide Metoclopramide is a dopamine D2 antagonist which has been used for treatment of a variety of gastrointestinal symptoms over the last thirty years. In various cou...
T7341 Diclofensine Diclofensine inhibits the uptake of serotonin, noradrenaline and dopamine.
T2793 Tetrahydropalmatine Tetrahydropalmatine is an active component isolated from corydalis, suppressing amygdaloid release of dopamine to inhibit an epileptic attack in rats.
T12352L Oxidopamine hydrobromide Oxidopamine hydrobromide is a neurotransmitter dopamine antagonist.
T10232 Acetophenazine dimaleate Acetophenazine dimaleate is an antipsychotic agent, effective in anxious depression.
TN1217 2'-O-Methylisoliquiritigenin 2'-O-Methylisoliquiritigenin, a compound synthesized by enzymes specifically induced in NR.
T8702 SKF-83566 SKF-83566 is a blood-brain permeable and orally active antagonist of D1-like dopamine receptor and a weaker competitive 5-HT2 receptor antagonist with Ki of 11 n...
T0302 Triflupromazine hydrochloride Triflupromazine hydrochloride, an antipsychotic medication, is Dopamine D1/D2 receptor antagonists.
T0137 Mirtazapine Mirtazapine is a tetracyclic antidepressant with a somewhat unique mechanism of action. Mirtazapine therapy can be associated with transient asymptomatic elevati...
T6647 Rotigotine- Rotigotine is a non-ergot dopamine receptor agonist used in the therapy of Parkinson disease and restless leg syndrome. Administered as a once-daily transdermal ...
T9540 Phenelzine Phenelzine is an antidepressant and mania drug, which is a monoamine oxidase inhibitor. Its antidepressant effect is similar to that of niacinamide. It can reduc...
T4S0779 D-tetrahydropalmatine D-Tetrahydropalmatine is a organic cation transporter 1 (OCT1) inhibitor, it can obviously inhibit the uptake of monocrotaline (MCT) in MDCK-hOCT1 cells and isol...
T12207 NEO 376 NEO 376 is a selective 5-HT1 receptor, GABA receptor and dopamine receptor modulator, showing anti-psychotic actively.
T4369 SCH-23390 hydrochloride SCH 23390 hydrochloride is an effective dopamine receptor antagonist, and for the D1(Ki=0.2 nM) and D5(Ki=0.3 nM).
T0351 Risperidone Risperidone is a selective blocker of dopamine D2 receptors and serotonin 5-HT2 receptors that act as an atypical antipsychotic agent.
T21667 FAUC-365 FAUC-365 is a D3 dopamine receptor agonist.
TQ0176 (-)-Isocorypalmine (-)-Isocorypalmine, a natural product isolated from Corydalis chaerophylla, has significant antifungal activity.
T0074L Chlorprothixene hydrochloride Chlorprothixene brings strong blocking effects by blocking the 5-HT2 D1, D2, D3, histamine H1, muscarinic and alpha1 adrenergic receptors. Chlorprothixene is a t...
T27677 JNJ-37822681 JNJ-37822681 is the first compound that allows the evaluation of the potential value of fast D(2) antagonism for the treatment of bipolar disorder and schizophre...
TQ0084 Lumateperone Tosylate Lumateperone Tosylate is a 5-HT2A receptor antagonist (Ki: 0.54 nM), a SERT blocker (Ki: 61 nM), a partial agonist of presynaptic D2 receptors and an antagonist ...
T21629 Loxapine Loxapine is a D2DR and D4DR inhibitor, serotonergic receptor antagonist and also a dibenzoxazepine anti-psychotic agent,used primarily in the treatment of schizo...
T11722 JNJ-37822681 dihydrochloride JNJ-37822681 has potential for the treatment of schizophrenia and bipolar disorder.JNJ-37822681 dihydrochloride is a potent, specific, centrally active, fast-dis...
T4494 CLOZAPINE N-OXIDE Clozapine N-oxide is a major metabolite of clozapine that can be detected in the earliest excretion time interval after clozapine administration [1]. It is produ...
T4008 Metergoline Metergoline is a dopamine agonist and serotonin antagonist. It has been used similarly to BROMOCRIPTINE as a dopamine agonist and also for migraine disorder ther...
T1222 Trifluoperazine dihydrochloride Trifluoperazine Dihydrochloride is a potent dopamine D2 receptor inhibitor used as an antipsychotic and an antiemetic.
T1105 Penfluridol Penfluridol is a highly potent antipsychotic.
T1322 Bendazol Bendazol is always used as the drug for hypertension and cerebral Angiospasm.
T22904 L-745870 trihydrochloride highly potent and selective D4 dopamine receptor antagonist
T14490 Talipexole dihydrochloride Talipexole dihydrochloride (B-HT 920 dihydrochloride) is a dopamine D2 receptor agonist, α2-adrenoceptor agonist and 5-HT3 receptor antagonist. It displays antiP...
T0338 Minaprine Minaprine is a reversible inhibitor of MAO-A, used in the treatment of various depressive states.
T10758L Centanafadine hydrochloride Centanafadine hydrochloride is a dual inhibitor of norepinephrine (NE)/dopamine (DA) transporter, also inhibits serotonin transporter (IC50s: 6 nM, 38 nM, and 83...
T14319 Aripiprazole Lauroxil Aripiprazole lauroxil is cleaved by body’s enzyme esterase to N-hydroxymethyl aripiprazole (plus lauric acid) and then to aripiprazole (plus formaldehyde), no to...
T12352 Oxidopamine hydrochloride Oxidopamine hydrochloride is an neurotransmitter dopamine antagonist.
T21446 Rotigotine Hydrochloride Rotigotine Hydrochloride, a dopamine receptor agonist prefering for D3 receptors over D1 and D2, has effective activity of anti-Parkinsonian. Racemic rotigotine ...
T12489 Pimethixene Pimethixene is a highly potent 5-HT1A, 5-HT2A, 5-HT2B, 5-HT2C, histamine H1, dopamine D2 and D4.4 as well as muscarinic M1 and M2 receptors antagonist(pKis of 7....
T2092 Amitifadine hydrochloride Amitifadine hydrochloride is a triple reuptake inhibitor (TRI) or serotonin-norepinephrine-dopamine reuptake inhibitor (SNDRI).
ABT 724 trihydrochloride
T22019
ABT 724 trihydrochloride 是一种有效的选择性 D4 受体激动剂(EC50 = 12.4 nM,14.3 nM 和 23.2 nM,分别对人、大鼠和雪貂)。 ABT-724 tri...
Dopamine hydrochloride
T1644
Dopamine is a naturally occurring catecholamine formed by decarboxylation of dihydroxyphenylalanine and a precursor of norepinephrine and epinephrine. Dopamine b...
Doxepin hydrochloride
T1540
Doxepin Hydrochloride is a dibenzoxepin tricyclic compound. It displays a range of pharmacological actions including maintaining adrenergic innervation. Its mech...
Methyldopa
T0505
Methyldopa, an alpha-adrenergic agonist (selective for α2-adrenergic receptors) psychoactive medicine, is served as an antihypertensive or sympatholytic.
Etilevodopa hydrochloride
T24047
Etilevodopa HCl is a prodrug of levodopa. It also has greater gastric solubility and significant brain penetration.
L-DOPA
T0848
Levodopa is an amino acid precursor of dopamine with antiparkinsonian properties. Levodopa is a prodrug that is converted to dopamine by DOPA decarboxylase and c...
Chlorprothixene
T0074
Chlorprothixene is a typical antipsychotic drug of the thioxanthene class, which was the first of the series to be synthesized.
WAY-100635 Maleate
T2631
WAY-100635 is a specific and effective 5-HT receptor antagonist (IC50=0.95 nM).
Metoclopramide hydrochloride hydrate
T8385
Metoclopramide hydrochloride hydrate is a dopamine D2 antagonist that is a drug used for digestive dysfunction. It acts as an anti-emetic
3-CPMT
T22508
dopamine uptake inhibitor
SCH-23390 maleate
T12865
SCH-23390 maleate is a potent and selective antagonist of dopamine D1-like receptor (1 and D5 receptor with Kis of 0.2 nM and 0.3 nM, respectively).
5-Benzyloxygramine
T35841
5-Benzyloxygramine is a N protein PPI orthosteric stabilizer that exhibits both antiviral and N-NTD protein-stabilizing activities[1]. 5-benzyloxygramine stabili...
Iloperidone
T1539
Iloperidone is an atypical antipsychotic agent that is used for treatment of schizophrenia.
Tetrahydropalmatine hydrochloride
T2917
Tetrahydropalmatine (THP) is an isoquinoline alkaloid found in several different plant species, mainly in the Corydalis genus (Yan Hu Suo). It is a potent muscle...
Metoclopramide
T4616
Metoclopramide is a dopamine D2 antagonist which has been used for treatment of a variety of gastrointestinal symptoms over the last thirty years. In various cou...
Diclofensine
T7341
Diclofensine inhibits the uptake of serotonin, noradrenaline and dopamine.
Tetrahydropalmatine
T2793
Tetrahydropalmatine is an active component isolated from corydalis, suppressing amygdaloid release of dopamine to inhibit an epileptic attack in rats.
Oxidopamine hydrobromide
T12352L
Oxidopamine hydrobromide is a neurotransmitter dopamine antagonist.
Acetophenazine dimaleate
T10232
Acetophenazine dimaleate is an antipsychotic agent, effective in anxious depression.
2'-O-Methylisoliquiritigenin
TN1217
2'-O-Methylisoliquiritigenin, a compound synthesized by enzymes specifically induced in NR.
SKF-83566
T8702
SKF-83566 is a blood-brain permeable and orally active antagonist of D1-like dopamine receptor and a weaker competitive 5-HT2 receptor antagonist with Ki of 11 n...
Triflupromazine hydrochloride
T0302
Triflupromazine hydrochloride, an antipsychotic medication, is Dopamine D1/D2 receptor antagonists.
Mirtazapine
T0137
Mirtazapine is a tetracyclic antidepressant with a somewhat unique mechanism of action. Mirtazapine therapy can be associated with transient asymptomatic elevati...
Rotigotine-
T6647
Rotigotine is a non-ergot dopamine receptor agonist used in the therapy of Parkinson disease and restless leg syndrome. Administered as a once-daily transdermal ...
Phenelzine
T9540
Phenelzine is an antidepressant and mania drug, which is a monoamine oxidase inhibitor. Its antidepressant effect is similar to that of niacinamide. It can reduc...
D-tetrahydropalmatine
T4S0779
D-Tetrahydropalmatine is a organic cation transporter 1 (OCT1) inhibitor, it can obviously inhibit the uptake of monocrotaline (MCT) in MDCK-hOCT1 cells and isol...
NEO 376
T12207
NEO 376 is a selective 5-HT1 receptor, GABA receptor and dopamine receptor modulator, showing anti-psychotic actively.
SCH-23390 hydrochloride
T4369
SCH 23390 hydrochloride is an effective dopamine receptor antagonist, and for the D1(Ki=0.2 nM) and D5(Ki=0.3 nM).
Risperidone
T0351
Risperidone is a selective blocker of dopamine D2 receptors and serotonin 5-HT2 receptors that act as an atypical antipsychotic agent.
FAUC-365
T21667
FAUC-365 is a D3 dopamine receptor agonist.
(-)-Isocorypalmine
TQ0176
(-)-Isocorypalmine, a natural product isolated from Corydalis chaerophylla, has significant antifungal activity.
Chlorprothixene hydrochloride
T0074L
Chlorprothixene brings strong blocking effects by blocking the 5-HT2 D1, D2, D3, histamine H1, muscarinic and alpha1 adrenergic receptors. Chlorprothixene is a t...
JNJ-37822681
T27677
JNJ-37822681 is the first compound that allows the evaluation of the potential value of fast D(2) antagonism for the treatment of bipolar disorder and schizophre...
lumateperone Tosylate
TQ0084
Lumateperone Tosylate is a 5-HT2A receptor antagonist (Ki: 0.54 nM), a SERT blocker (Ki: 61 nM), a partial agonist of presynaptic D2 receptors and an antagonist ...
Loxapine
T21629
Loxapine is a D2DR and D4DR inhibitor, serotonergic receptor antagonist and also a dibenzoxazepine anti-psychotic agent,used primarily in the treatment of schizo...
JNJ-37822681 dihydrochloride
T11722
JNJ-37822681 has potential for the treatment of schizophrenia and bipolar disorder.JNJ-37822681 dihydrochloride is a potent, specific, centrally active, fast-dis...
CLOZAPINE N-OXIDE
T4494
Clozapine N-oxide is a major metabolite of clozapine that can be detected in the earliest excretion time interval after clozapine administration [1]. It is produ...
Metergoline
T4008
Metergoline is a dopamine agonist and serotonin antagonist. It has been used similarly to BROMOCRIPTINE as a dopamine agonist and also for migraine disorder ther...
Trifluoperazine dihydrochloride
T1222
Trifluoperazine Dihydrochloride is a potent dopamine D2 receptor inhibitor used as an antipsychotic and an antiemetic.
Penfluridol
T1105
Penfluridol is a highly potent antipsychotic.
Bendazol
T1322
Bendazol is always used as the drug for hypertension and cerebral Angiospasm.
L-745870 trihydrochloride
T22904
highly potent and selective D4 dopamine receptor antagonist
Talipexole dihydrochloride
T14490
Talipexole dihydrochloride (B-HT 920 dihydrochloride) is a dopamine D2 receptor agonist, α2-adrenoceptor agonist and 5-HT3 receptor antagonist. It displays anti...
Minaprine
T0338
Minaprine is a reversible inhibitor of MAO-A, used in the treatment of various depressive states.
Centanafadine hydrochloride
T10758L
Centanafadine hydrochloride is a dual inhibitor of norepinephrine (NE)/dopamine (DA) transporter, also inhibits serotonin transporter (IC50s: 6 nM, 38 nM, and 83...
Aripiprazole Lauroxil
T14319
Aripiprazole lauroxil is cleaved by body’s enzyme esterase to N-hydroxymethyl aripiprazole (plus lauric acid) and then to aripiprazole (plus formaldehyde), no ...
Oxidopamine hydrochloride
T12352
Oxidopamine hydrochloride is an neurotransmitter dopamine antagonist.
Rotigotine Hydrochloride
T21446
Rotigotine Hydrochloride, a dopamine receptor agonist prefering for D3 receptors over D1 and D2, has effective activity of anti-Parkinsonian. Racemic rotigotine ...
Pimethixene
T12489
Pimethixene is a highly potent 5-HT1A, 5-HT2A, 5-HT2B, 5-HT2C, histamine H1, dopamine D2 and D4.4 as well as muscarinic M1 and M2 receptors antagonist(pKis of 7....
Amitifadine hydrochloride
T2092
Amitifadine hydrochloride is a triple reuptake inhibitor (TRI) or serotonin-norepinephrine-dopamine reuptake inhibitor (SNDRI).
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