AChR

An acetylcholine receptor (abbreviated AChR) is an integral membrane protein that responds to the binding of acetylcholine, a neurotransmitter.

Cat. No.	Product name	CAS No.	Purity
T21532	Anisodamine	55869-99-3	98%
T21532	6-beta-Hydroxyhyoscyamine and 7 beta-hydroxyhyoscyamine exhibit similar affinities at the muscarinic receptor as scopolamine and atropine.
T62769	Tribendimidine	115103-15-6	98%
T62769	Tribendimidine is an orally active and broad-spectrum anthelmintic agent. Tribendimidine exhibits particularly high activity against A. lumbricoides and N. ameri...
TN3287	8-Lavandulylkaempferol	883859-83-4	98%
TN3287	8-Lavandulylkaempferol exhibits significant inhibitory effects with IC(50) values of 7.10 and 8.11 microM for butyrylcholinesterase and acetylcholinesterase, res...
T5476	MAChr-in-1	119391-56-9	98%
T5476	mAChR-IN-1 is muscarinic cholinergic receptor(mAChR) antagonist (IC50=17 nM).
T10914	Cyclodrine hydrochloride	78853-39-1	98%
T10914	Cyclone hydrochloride is a cholinergic (muscarinic, nicotinic) (mAChR and nAChR) receptor antagonist.
TN3744	Cyclomorusin	62596-34-3	98%
TN3744	Cyclomorusin exhibits competitive inhibition toward monophenolase activity of mushroom tyrosinase, the IC50 value of 0.092 microM. It evokes the stimulation of s...
TN2067	Picfeltarraegenin X	1391826-61-1	98%
TN2067	Picfeltarraenin X shows stronger AChE inhibition than the known AChE inhibitor Tacrine.
T12446	Phenserine	101246-66-6	98%
T12446	Phenserine is a derivative of Physostigmine and is annoncompetitive, long-acting and selective inhibitor of AChE.
T61233	Penehyclidine hydrochloride	151937-76-7	98%
T61233	Penehyclidine hydrochloride is an M1 and M3 antagonist and activates NF-κB in lung tissue. Penehyclidine hydrochloride inhibits the release of inflammatory facto...
T12868	Sch412348	377727-26-9	98%
T12868	Sch412348 is a potent competitive the human adenosine A2A receptor antagonist with Ki of 0.6 nM and has >1000-fold selectivity over all other adenosine receptors...
T0218	Biperiden	514-65-8	98%
T0218	Biperiden is a muscarinic antagonist that has effects in both the central and peripheral nervous systems. It has been used in the treatment of arteriosclerotic, ...
T7224	Anabasine	494-52-0	98%
T7224	Anabasine is a nicotine analog that is an alkaloid found in tree tobacco (Nicotiana glauca). Anabasine has been used as an industrial insecticide and, since it i...
T16563	Pozanicline	161417-03-4	98%
T16563	Pozanicline reverses nicotine withdrawal-induced cognitive deficits, may be an effective component of novel therapeutic strategies for nicotine addiction. Pozani...
TL0018	Lobelin	90-69-7	98%
TL0018	Inhalation challenge with capsaicin and rapid intravenous injection of Lobelin and alinamin indicated that peripheral c-fiber receptors were involved in the indu...
T1484	Perindoprilat	95153-31-4	98%
T1484	Perindoprilat is an angiotensin-converting enzyme inhibitor.
T22486	Vesamicol hydrochloride	120447-62-3	98%
T22486	Vesamicol hydrochloride is a acetylcholine transport inhibitor.
T19623	α-Muricholic acid	2393-58-0	98%
T19623	α-Muricholic acid is the most abundant primary bile acid in rodents.
TN5193	Tubotaiwine	6711-69-9	98%
TN5193	Tubotaiwine shows selective activity against L. infantum. Tubotaiwine and apparicine have affinity for adenosine receptors in the micromolar range and also have ...
T12107	MRS-3777 hemioxalate	1186195-57-2	98%
T12107	MRS-3777 hemioxalate is a selective antagonist of adenosine A3 receptor .
TQ0304	Metixene hydrochloride hydrate	7081-40-5	98%
TQ0304	Metixene is an anticholinergic antiparkinsonian agent, potently inhibits the binding of quinuclidinyl to the muscarinic receptor in rat brain cortical tissue (IC...