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AChR

An acetylcholine receptor (abbreviated AChR) is an integral membrane protein that responds to the binding of acetylcholine, a neurotransmitter.
Cat. No. Product name CAS No. Purity Chemical Structure
TN2217 Sophoflavescenol 216450-65-6 99.65%
Sophoflavescenol is a mixed inhibitor of PDE5 with a K(i) value of 0.005 microM. Sophoflavescenol has antioxidant, anti-inflammatory, and apoptotic effects , the...
TN1798 Isorosmanol 93780-80-4 98.85%
Isorosmanol possesses antioxidant, neuroprotective and neurotrophic effects, it might be useful in ageing disorders such as the declining of cognitive functions ...
T0346 Camylofine 54-30-8 98%
Camylofin is an antimuscarinic, used for relaxing smooth muscle.
TN1519 (S)-Coclaurine 486-39-5 97.72%
(S)-Coclaurine is an antagonist of nAChR isolated from Sarcopetalum harveyanum.
T8702 SKF-83566 99295-33-7 95.00%
SKF-83566 is a blood-brain permeable and orally active antagonist of D1-like dopamine receptor and a weaker competitive 5-HT2 receptor antagonist with Ki of 11 n...
T68019 Ursulcholic acid 88426-32-8 100%
Ursulcholic acid is a water-soluble anticholinergic compound.
T1236 Pentolinium Tartrate 52-62-0
A nicotinic antagonist that has been used as a ganglionic blocking agent in hypertension.
T0218 Biperiden 514-65-8
Biperiden is a muscarinic antagonist that has effects in both the central and peripheral nervous systems. It has been used in the treatment of arteriosclerotic, ...
T13129 Terodiline hydrochloride 7082-21-5 98%
Terodiline hydrochloride is an antagonist of M1-selective muscarinic receptor (mAChR)(Kbs of 15, 160, 280, and 198 nM in rabbit vas deferens (M1), atria (M2), bl...
T6721 Vinblastine 865-21-4 98%
Vinblastine inhibits microtubule formation and suppresses nAChR activity with IC50 of 8.9 μM, used to treat certain kinds of cancer.
TN4837 Pseudotaraxasterol 464-98-2 98%
Pseudotaraxasterol shows cytotoxic activity against MOLT-4 cells.
TN3696 Conodurine 2665-57-8 98%
Conodurine shows leishmanicidal and antibacterial activities, it shows inhibition activity for acetyl (AChE) and butyrylcholinesterase (BuChE).
T7224 Anabasine 494-52-0 98%
Anabasine is a nicotine analog that is an alkaloid found in tree tobacco (Nicotiana glauca). Anabasine has been used as an industrial insecticide and, since it i...
TN1559 Dehydrodicentrine 19843-03-9 98%
Dehydrodicentrine showed strong acetylcholinesterase (AChE) inhibitory effects with the IC50 value of 2.98 μM.
T12020 Metixene hydrochloride 1553-34-0 98%
Metixene hydrochloride is an anticholinergic antiparkinsonian agent.
TN1645 Flavokawain C 56798-34-6 98%
Flavokawain C is a melanogenesis inhibitor, it inhibited melanogenesis with IC50 values of 6.9 μM. Flavokawain C has anti-tumor activity, it inhibited cell cycle...
TN1653 Fustin 20725-03-5 98%
Fustin shows protective effects on 6-hydroxydopamine-induced neuronal cell death.
TN3380 Alloisoimperatorin 35214-83-6 98%
Alloisoimperatorin is a candidate of AChE inhibitors, it displays potent antioxidant effects against the DPPH radical and against renal epithelial cell injury by...
T13713 GP531 142344-87-4 98%
GP531 is a second-generation adenosine regulating agent. It is pharmacologically silent under basal conditions but increases localized endogenous adenosine durin...
TN2505 1,5-Diphenylpentan-1-one 39686-51-6 98%
1,5-Diphenylpentan-1-one shows poor insecticidal and acetylcholinesterase inhibitory activities.
Sophoflavescenol
TN2217
Sophoflavescenol is a mixed inhibitor of PDE5 with a K(i) value of 0.005 microM. Sophoflavescenol has antioxidant, anti-inflammatory, and apoptotic effects , the...
Isorosmanol
TN1798
Isorosmanol possesses antioxidant, neuroprotective and neurotrophic effects, it might be useful in ageing disorders such as the declining of cognitive functions ...
Camylofine
T0346
Camylofin is an antimuscarinic, used for relaxing smooth muscle.
(S)-Coclaurine
TN1519
(S)-Coclaurine is an antagonist of nAChR isolated from Sarcopetalum harveyanum.
SKF-83566
T8702
SKF-83566 is a blood-brain permeable and orally active antagonist of D1-like dopamine receptor and a weaker competitive 5-HT2 receptor antagonist with Ki of 11 n...
Ursulcholic acid
T68019
Ursulcholic acid is a water-soluble anticholinergic compound.
Pentolinium Tartrate
T1236
A nicotinic antagonist that has been used as a ganglionic blocking agent in hypertension.
Biperiden
T0218
Biperiden is a muscarinic antagonist that has effects in both the central and peripheral nervous systems. It has been used in the treatment of arteriosclerotic, ...
Terodiline hydrochloride
T13129
Terodiline hydrochloride is an antagonist of M1-selective muscarinic receptor (mAChR)(Kbs of 15, 160, 280, and 198 nM in rabbit vas deferens (M1), atria (M2), bl...
Vinblastine
T6721
Vinblastine inhibits microtubule formation and suppresses nAChR activity with IC50 of 8.9 μM, used to treat certain kinds of cancer.
Pseudotaraxasterol
TN4837
Pseudotaraxasterol shows cytotoxic activity against MOLT-4 cells.
Conodurine
TN3696
Conodurine shows leishmanicidal and antibacterial activities, it shows inhibition activity for acetyl (AChE) and butyrylcholinesterase (BuChE).
Anabasine
T7224
Anabasine is a nicotine analog that is an alkaloid found in tree tobacco (Nicotiana glauca). Anabasine has been used as an industrial insecticide and, since it i...
Dehydrodicentrine
TN1559
Dehydrodicentrine showed strong acetylcholinesterase (AChE) inhibitory effects with the IC50 value of 2.98 μM.
Metixene hydrochloride
T12020
Metixene hydrochloride is an anticholinergic antiparkinsonian agent.
Flavokawain C
TN1645
Flavokawain C is a melanogenesis inhibitor, it inhibited melanogenesis with IC50 values of 6.9 μM. Flavokawain C has anti-tumor activity, it inhibited cell cycle...
Fustin
TN1653
Fustin shows protective effects on 6-hydroxydopamine-induced neuronal cell death.
Alloisoimperatorin
TN3380
Alloisoimperatorin is a candidate of AChE inhibitors, it displays potent antioxidant effects against the DPPH radical and against renal epithelial cell injury by...
GP531
T13713
GP531 is a second-generation adenosine regulating agent. It is pharmacologically silent under basal conditions but increases localized endogenous adenosine durin...
1,5-Diphenylpentan-1-one
TN2505
1,5-Diphenylpentan-1-one shows poor insecticidal and acetylcholinesterase inhibitory activities.
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