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AChR

An acetylcholine receptor (abbreviated AChR) is an integral membrane protein that responds to the binding of acetylcholine, a neurotransmitter.
Cat. No. Product name CAS No. Purity Chemical Structure
T21532 Anisodamine 55869-99-3 98%
6-beta-Hydroxyhyoscyamine and 7 beta-hydroxyhyoscyamine exhibit similar affinities at the muscarinic receptor as scopolamine and atropine.
T62769 Tribendimidine 115103-15-6 98%
Tribendimidine is an orally active and broad-spectrum anthelmintic agent. Tribendimidine exhibits particularly high activity against A. lumbricoides and N. ameri...
TN3287 8-Lavandulylkaempferol 883859-83-4 98%
8-Lavandulylkaempferol exhibits significant inhibitory effects with IC(50) values of 7.10 and 8.11 microM for butyrylcholinesterase and acetylcholinesterase, res...
T5476 MAChr-in-1 119391-56-9 98%
mAChR-IN-1 is muscarinic cholinergic receptor(mAChR) antagonist (IC50=17 nM).
T10914 Cyclodrine hydrochloride 78853-39-1 98%
Cyclone hydrochloride is a cholinergic (muscarinic, nicotinic) (mAChR and nAChR) receptor antagonist.
TN3744 Cyclomorusin 62596-34-3 98%
Cyclomorusin exhibits competitive inhibition toward monophenolase activity of mushroom tyrosinase, the IC50 value of 0.092 microM. It evokes the stimulation of s...
TN2067 Picfeltarraegenin X 1391826-61-1 98%
Picfeltarraenin X shows stronger AChE inhibition than the known AChE inhibitor Tacrine.
T12446 Phenserine 101246-66-6 98%
Phenserine is a derivative of Physostigmine and is annoncompetitive, long-acting and selective inhibitor of AChE.
T61233 Penehyclidine hydrochloride 151937-76-7 98%
Penehyclidine hydrochloride is an M1 and M3 antagonist and activates NF-κB in lung tissue. Penehyclidine hydrochloride inhibits the release of inflammatory facto...
T12868 Sch412348 377727-26-9 98%
Sch412348 is a potent competitive the human adenosine A2A receptor antagonist with Ki of 0.6 nM and has >1000-fold selectivity over all other adenosine receptors...
T0218 Biperiden 514-65-8 98%
Biperiden is a muscarinic antagonist that has effects in both the central and peripheral nervous systems. It has been used in the treatment of arteriosclerotic, ...
T7224 Anabasine 494-52-0 98%
Anabasine is a nicotine analog that is an alkaloid found in tree tobacco (Nicotiana glauca). Anabasine has been used as an industrial insecticide and, since it i...
T16563 Pozanicline 161417-03-4 98%
Pozanicline reverses nicotine withdrawal-induced cognitive deficits, may be an effective component of novel therapeutic strategies for nicotine addiction. Pozani...
TL0018 Lobelin 90-69-7 98%
Inhalation challenge with capsaicin and rapid intravenous injection of Lobelin and alinamin indicated that peripheral c-fiber receptors were involved in the indu...
T1484 Perindoprilat 95153-31-4 98%
Perindoprilat is an angiotensin-converting enzyme inhibitor.
T22486 Vesamicol hydrochloride 120447-62-3 98%
Vesamicol hydrochloride is a acetylcholine transport inhibitor.
T19623 α-Muricholic acid 2393-58-0 98%
α-Muricholic acid is the most abundant primary bile acid in rodents.
TN5193 Tubotaiwine 6711-69-9 98%
Tubotaiwine shows selective activity against L. infantum. Tubotaiwine and apparicine have affinity for adenosine receptors in the micromolar range and also have ...
T12107 MRS-3777 hemioxalate 1186195-57-2 98%
MRS-3777 hemioxalate is a selective antagonist of adenosine A3 receptor .
TQ0304 Metixene hydrochloride hydrate 7081-40-5 98%
Metixene is an anticholinergic antiparkinsonian agent, potently inhibits the binding of quinuclidinyl to the muscarinic receptor in rat brain cortical tissue (IC...
Anisodamine
T21532
6-beta-Hydroxyhyoscyamine and 7 beta-hydroxyhyoscyamine exhibit similar affinities at the muscarinic receptor as scopolamine and atropine.
Tribendimidine
T62769
Tribendimidine is an orally active and broad-spectrum anthelmintic agent. Tribendimidine exhibits particularly high activity against A. lumbricoides and N. ameri...
8-Lavandulylkaempferol
TN3287
8-Lavandulylkaempferol exhibits significant inhibitory effects with IC(50) values of 7.10 and 8.11 microM for butyrylcholinesterase and acetylcholinesterase, res...
mAChr-in-1
T5476
mAChR-IN-1 is muscarinic cholinergic receptor(mAChR) antagonist (IC50=17 nM).
Cyclodrine hydrochloride
T10914
Cyclone hydrochloride is a cholinergic (muscarinic, nicotinic) (mAChR and nAChR) receptor antagonist.
Cyclomorusin
TN3744
Cyclomorusin exhibits competitive inhibition toward monophenolase activity of mushroom tyrosinase, the IC50 value of 0.092 microM. It evokes the stimulation of s...
Picfeltarraegenin X
TN2067
Picfeltarraenin X shows stronger AChE inhibition than the known AChE inhibitor Tacrine.
Phenserine
T12446
Phenserine is a derivative of Physostigmine and is annoncompetitive, long-acting and selective inhibitor of AChE.
Penehyclidine hydrochloride
T61233
Penehyclidine hydrochloride is an M1 and M3 antagonist and activates NF-κB in lung tissue. Penehyclidine hydrochloride inhibits the release of inflammatory facto...
Sch412348
T12868
Sch412348 is a potent competitive the human adenosine A2A receptor antagonist with Ki of 0.6 nM and has >1000-fold selectivity over all other adenosine receptors...
Biperiden
T0218
Biperiden is a muscarinic antagonist that has effects in both the central and peripheral nervous systems. It has been used in the treatment of arteriosclerotic, ...
Anabasine
T7224
Anabasine is a nicotine analog that is an alkaloid found in tree tobacco (Nicotiana glauca). Anabasine has been used as an industrial insecticide and, since it i...
Pozanicline
T16563
Pozanicline reverses nicotine withdrawal-induced cognitive deficits, may be an effective component of novel therapeutic strategies for nicotine addiction. Pozani...
Lobelin
TL0018
Inhalation challenge with capsaicin and rapid intravenous injection of Lobelin and alinamin indicated that peripheral c-fiber receptors were involved in the indu...
Perindoprilat
T1484
Perindoprilat is an angiotensin-converting enzyme inhibitor.
Vesamicol hydrochloride
T22486
Vesamicol hydrochloride is a acetylcholine transport inhibitor.
α-Muricholic acid
T19623
α-Muricholic acid is the most abundant primary bile acid in rodents.
Tubotaiwine
TN5193
Tubotaiwine shows selective activity against L. infantum. Tubotaiwine and apparicine have affinity for adenosine receptors in the micromolar range and also have ...
MRS-3777 hemioxalate
T12107
MRS-3777 hemioxalate is a selective antagonist of adenosine A3 receptor .
Metixene hydrochloride hydrate
TQ0304
Metixene is an anticholinergic antiparkinsonian agent, potently inhibits the binding of quinuclidinyl to the muscarinic receptor in rat brain cortical tissue (IC...
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