T13592 |
Calf thymus DNA
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DNA from calf thymus, Thymonucleic acid |
DNA/RNA Synthesis
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Calf thymus DNA 是一种从牛胸腺中提取出来的高质量双链模板DNA,可广泛应用于DNA 结合抗癌剂和调节DNA 结构和功能的DNA 结合剂的研究。 |
T31554 |
DNA-Spermidine
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DA 51,DA-51,DA51,DNA Spermidine |
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DNA-spermidine influences the activity of restricted endonuclease from several bacterial species. |
T74337 |
DNA crosslinker 1 dihydrochloride
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DNA crosslinker 1 (dihydrochloride) 是一种有效的DNA 小沟结合剂,与 DNA 的结合亲和力 (ΔTm) 为 1.1 °C。DNA crosslinker 1 (dihydrochloride) 可用于抗... |
T74339 |
DNA crosslinker 3 dihydrochloride
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DNA crosslinker 3 (dihydrochloride) (compound 1) 是一种DNA 小沟结合剂,与 DNA 的结合亲和力 (ΔTm) 为 1.4 °C。DNA crosslinker 3 (dihydrochlo... |
T74340 |
DNA crosslinker 4 dihydrochloride
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DNA crosslinker 4 (dihydrochloride) 是一种有效的 DNA 小沟结合剂。DNA crosslinker 4 (dihydrochloride) 对癌细胞 NCI-H460、A2780 和 MCF-7 有一定... |
T63681 |
DNA Gyrase-IN-1
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DNA Gyrase-IN-1 是有效的、选择性的 DNA 促旋酶抑制剂 (IC50: 2.6 μM)。DNA Gyrase-IN-1 能够较好的抑制结核分枝杆菌 (Mtb) 的活性 (MIC: 0.49 μM)。DNA Gyrase-IN... |
T61751 |
DNA-PK-IN-3
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DNA-PK-IN-3 is a highly potent inhibitor of DNA-PK. This compound exerts a synergistic effect when combined with radioth... |
T74848 |
DNA Gyrase-IN-6
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Antibacterial agent 138 是细菌 DNA 促旋酶和拓扑异构酶 IV 的苯并噻唑抑制剂。Antibacterial agent 138 表现出良好的溶解度和血浆蛋白结合。Antibacterial agent 138 对... |
T61937 |
DNA Gyrase-IN-3
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DNA Gyrase-IN-3 (Compound 28) 是细菌DNA 旋转酶 B (bacterial DNA gyrase B) 抑制剂。DNA Gyrase-IN-3抑制大肠杆菌DNA 旋转酶的 IC50为5.41-15.64 μM... |
T61857 |
DNA-PK-IN-4
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DNA-PK-IN-4 (WO2021209055A1, compound 27), an imidazolinone derivative compound, is a highly effective inhibitor of DNA-... |
T74338 |
DNA crosslinker 2 dihydrochloride
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DNA crosslinker 2 (dihydrochloride) 是一种有效的 DNA 小沟结合剂,与 DNA 的结合亲和力 (ΔTm) 为 1.2 °C。DNA crosslinker 2 (dihydrochloride) 对癌细... |
T62191 |
DNA-PK-IN-5
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DNA-PK-IN-5 是一种 DNA-PK 的有效抑制剂。DNA-PK-IN-5 能够抑制 DNA-PKcs 活性,明显降低肿瘤 DNA 修复,并诱导细胞凋亡。DNA-PK-IN-5 能够提高肿瘤组织对放疗的敏感性,克服耐药问题,提高对多... |
T62034 |
DNA-PK-IN-7
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DNA-PK-IN-7 是有效的 DNA-PK 抑制剂,IC50为 1 nM (WO2021104277A1, compound 5)。 |
T63395 |
DNA Gyrase-IN-5
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DNA Gyrase-IN-5 是 DNA gyrase 的有效抑制剂 (IC50: 0.10 μM),对野生型和耐药株均有抗细菌(antibacterial)作用。 |
T64012 |
DNA gyrase B-IN-1
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DNA gyrase B-IN-1 是 DNA gyrase B 的有效抑制剂,表现出良好的结合亲和力和稳定性。DNA gyrase B-IN-1 能够抑制 P. aeruginosa/i> DNA gyrase B (IC50: 2.2 ... |
T61633 |
DNA-PK-IN-2
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DNA-PK-IN-2 is a highly effective inhibitor of DNA-dependent protein kinase (DNA-PK), which is a complex enzyme composed... |
T62648 |
DNA-PK-IN-1
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DNA-PK-IN-1 是一种 DNA-PK 的有效抑制剂。DNA 依赖性蛋白激酶 (DNA-PK) 是一种由 Ku70/Ku80 异二聚体和 DNA 依赖性蛋白激酶催化亚基 (DNA-PKcs) 组成的 DNA-PK 酶复合物。DNA-P... |
T61533 |
DNA-PK-IN-9
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DNA-PK-IN-9 (also known as compound YK6) is a highly potent inhibitor of DNA-dependent protein kinase (DNA-PK), displayi... |
T63442 |
DNA Gyrase-IN-2
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DNA Gyrase-IN-2 是细菌 DNA 促旋酶 B 抑制剂,能作用于大肠杆菌 DNA 促旋酶(IC50: 3.29-10.49 μM)和结核分枝杆菌 DNA 促旋酶(IC50: 4.41-5.61 μM),表现出抗菌和抗结核作用。 |
T60961 |
LANA-DNA-IN-1
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LANA-DNA-IN-1 是 LANA-DNA 的有效抑制剂,对 LBS2、LBS1 和 LBS3 的 IC50值分别为 8 μM、9μM 和 8μM。 LANA-DNA-IN-1 对野生型 LANA 显示出 53 μM 的 IC50值。... |