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Results for "a-1" in TargetMol Product Catalog
  • Inhibitor Products
    17422
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    2215
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Cyt-PTPε Inhibitor-1
T10927428478-94-8In house
Cyt-PTPε Inhibitor-1 (A Inhibitor-1) is an inhibitor of cytosolic protein tyrosine phosphatase ε. Cyt-PTPε Inhibitor-1 blocks the dephosphorylation of c-Src and exhibits anti-osteoclastic activity.
  • $58
In Stock
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[DPro10] Dynorphin A (1-11)acetate,porcine
T76341L
[DPro10] Dynorphin A (1-11)acetate,porcine is a highly potent κ-opioid receptor agonist with a Ki value of 0.13 nM. [DPro10] Dynorphin A (1-11), porcine is an n-alkylated derivative with analgesic activity.
  • $55
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Pulsatilla saponin H
TN211968027-14-5
Pulsatilla saponin H is a natural product isolated from the Roots of Pulsatilla koreana.
  • $389
In Stock
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Dynorphin A 1-10 acetate(79994-24-4 free base)
TP1813L
Dynorphin A (1-10) acetate is an endogenous opioid neuropeptide, binds to extracellular loop 2 of the κ-opioid receptor. Dynorphin A (1-10) also blocks NMDA-activated current with an IC50 of 42.0 μM.
  • $101
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(+/-)-Longamide
TN7157219783-00-3
(+/-)-Longamide (6,7-dibromo-4-hydroxy-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-1-one) is a marine derived natural products found in Sponge Homaxinella sp.
  • $195
In Stock
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Porcine dynorphin A(1-13) acetate
TP1179L
Porcine dynorphin A(1-13) acetate (Dynorphin A Porcine Fragment 1-13 acetate) is a potent, endogenous κ opioid receptor agonist and is antinociceptive at physiological concentrations. Exposure to dynorphin A (1-13) causes acute increases in [Ca2+]i in individual neurons similar to increases seen with acute NMDA treatment.
  • $68
In Stock
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QTY
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Angiotensin 1/2 + A (2 - 8) Acetate
T21708L
Angiotensin 1/2 + A (2 - 8) Acetate is a Vasoconstrictor.
  • $68
In Stock
Size
QTY
Levofloxacin Hydrochloride Impurity A
T11007L2254176-11-7
Levofloxacin Hydrochloride Impurity A I, one of the quinolones, has a broad spectrum of antibacterial action.
  • $148
In Stock
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QTY
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Mukanadin C
TN71481839104-78-7
Mukanadin C (7-bromo-4-hydroxy-3,4-dihydro-2H-pyrrolo[1,2-a]pyrazin-1-one) is a marine derived natural products found in Stylissa carteri.
  • $195
In Stock
Size
QTY
SPOP-IN-6b
T169222136270-20-5In house
SPOP-IN-6b is an effective inhibitor of speckle-type POZ protein (SPOP) with an IC50 of 3.58 μM and can be used in stuides about the treatment of renal cancer.
  • $96
In Stock
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QTY
A-176120 ammonium
T26469L In house
A-176120 ammonium is a novel farnesyl pyrophosphate analog with antitumor and antiangiogenic properties and inhibits farnesyltransferase activity.
  • $397
In Stock
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Dorsomorphin dihydrochloride
T61461219168-18-9
Dorsomorphin dihydrochloride (BML-275 2HCl) is a potent, selective and ATP-competitive AMPK inhibitor (Ki: 109 nM) and does not exhibit significant activity on structurally related kinases.
  • $30
In Stock
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TargetMol | Citations Cited
Dynorphin A (1-13) amide
T8251979515-34-7
Dynorphin A (1-13) amide, an endogenous opioid peptide, counteracts the analgesic effects of morphine [1].
  • Inquiry Price
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Pulsatilloside E
TN2117366814-43-9
Pulsatilloside E (Pulchinenoside E) is a natural product isolated from the roots of Pulsatilla chinensis (Ranunculaceae).
  • $115
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Aclerastide
T26554227803-63-6
Aclerastide is an angiotensin receptor agonist. Administration of Aclerastide reduced fibrosis and scarring in the healing wounds. This action was more pronounced with longer administration of the peptide after injury. The action of this peptide was block
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3-O-β-D-Glucopyranosyl(1→2)-[a-Lrhamnopyranosyl(1→3)]-β-D-glucopyranosyl 28-O-β-D-glucuronopyranoside
T83344110081-91-9
3-O-β-D-Glucopyranosyl(1→2)-[α-L-rhamnopyranosyl(1→3)]-β-D-glucopyranosyl 28-O-β-D-glucuronopyranoside is a saponin compound extracted from Polaskia chichipe Backbg. It demonstrates an 84.2% inhibitory activity on melanin biosynthesis at a concentration of 100μM in B16 melanoma cells[1].
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Ceramide 1 A
T30797179186-48-2
Ceramide 1 A is a waxy lipid compound that is a lipid in the top skin layer. It has a special molecular structure because it contains a linoleic acid linked to a long chain omega-hydroxy acid.
  • $1,520
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Cyclosporin A-Derivative 1 Free base
TP1405286852-20-8
Cyclosporin A-Derivative 1 (Free base) is a crystalline intermediate derived from the opening of cyclosporin A.
  • $121
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Avenacin A 1
T3022290547-90-3
Avenacin A 1 is a biochemical.
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Melan-A/MART-1 analog
T81825204060-45-7
[Leu27]-Melan-A, MART-1 (26-35), is a biologically active peptide modified by substituting leucine for alanine at position 27, which enhances its HLA-A*0201 binding, immunogenicity, and antigenicity compared to the natural peptide. Pyroglutamyl (pGlu) peptides, arising from the spontaneous cyclization of glutamine (Q) or glutamic acid (E) at the N-terminus, are a recognized subset of peptides that may confer increased stability due to the hydrophobic γ-lactam ring of pGlu. These pGlu peptides are typically included during peptide purity assessments in HPLC analysis.
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D-MoDE-A (1)
T825372378837-67-1
D-MoDE-A (1) is a bifunctional small molecule that facilitates extracellular protein degradation via the asialoglycoprotein receptor (ASGPR).
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[DPro10] Dynorphin A (1-11), porcine
T7634194596-26-6
[DPro10] Dynorphin A (1-11), porcine, an N-Alkylated derivative, serves as a potent κ-opioid receptor agonist with a Ki value of 0.13 nM, exhibiting analgesic properties [1] [2].
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[DAla2] Dynorphin A (1-9) (porcine)
T8350595673-38-4
[DAla2] Dynorphin A (1-9) (porcine) is a dynorphin utilized in research related to analgesic, addiction, and depression studies.
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KRAS G12C mutant protein inhibitor A-1
T778052658538-04-4
KRAS G12C mutant protein inhibitor A-1 can be used in studies about Ras.
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Dynorphin A (1-10) TFA(79994-24-4,free)
TP1423
Dynorphin A (1-10) (TFA), an endogenous opioid neuropeptide, binds in the transmembrane domain of the κ-receptor.
  • $72
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Kadsurin A analogue-1
T81993155551-59-0
Kadsurin A Analogue-1 (Compound 8), a lignan, can be extracted from Piper argyrophylum [1].
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Thaxtomin A
T34834122380-18-1
Thaxtomin A is a plant toxin that causes the death of plant cells.
  • $248
35 days
Size
QTY
TargetMol | Inhibitor Sale
a-Bag Cell Peptide (1-8)
T8322087549-53-9
α-Bag Cell Peptide (1-8) is an NH2-terminal fragment of α-bag cell peptide that inhibits LUQ (left upper quadrant) neurons and the depolarization of bag cells [1].
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a-Bag Cell Peptide (1-7)
T8322187549-54-0
α-Bag Cell Peptide (1-7) is an amino-terminal fragment of the α-bag cell peptide that possesses the ability to inhibit neurons in the left upper quadrant (LUQ) and prevent the depolarization of the bag cells [1].
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A1B11
T235921602731-56-5
A1B11 is a selective SIRT2 inhibitor.
  • $2,270
10-14 weeks
Size
QTY
3'-Rhamnopiericidin A(1)
T29419131622-62-3
3'-Rhamnopiericidin A(1) is a piericidin rhamnoside from Streptomyces.
  • Inquiry Price
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[DAla2, DArg6] Dynorphin A, (1-13) (porcine)
T7633775921-88-9
[DAla2, DArg6] Dynorphin A, (1-13) (porcine) (DADAD), a dynorphin1-13 (DYN) derivative extracted from porcine pituitary, exhibits high potency at peripheral opioid receptors GPI and MVD. Despite rapid in vivo degradation of DYN, this compound shows increased resistance to enzymatic cleavage, enhancing its stability against peptide-degrading enzymes [1].
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Cecropin A (1-7)-Melittin A (2-9)
T76468157606-25-2
Cecropin A (1-7)-Melittin A (2-9) is an antimicrobial peptide that exhibits broad-spectrum antimicrobial activity against both Gram-positive and Gram-negative aerobic bacteria, in addition to antimalarial properties. Notably, it does not possess the adverse hemolytic effects commonly associated with bee venom peptides [1].
  • Inquiry Price
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Ajugamarin A 1
T2978778798-40-0
Ajugamarin A 1 is a Neoclerodane diterpenoid.
  • $1,520
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(N-Me-Tyr1,N-Me-Arg7,D-Leu-NHEt8)-Dynorphin A (1-8)
T76631103613-84-9
E-2078, known chemically as (N-Me-Tyr1,N-Me-Arg7,D-Leu-NHEt8)-Dynorphin A (1-8), is a stable analog of Dynorphin A (1–8) and functions as a kappa opioid receptor (KOR) agonist [1].
  • Inquiry Price
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3,8-Dihydroxy-1-methylanthraquinone-2-carboxylic a
T12438069119-31-9
3,8-Dihydroxy-1-methylanthraquinone-2-carboxylic a is a useful organic compound for research related to life sciences. The catalog number is T124380 and the CAS number is 69119-31-9.
  • Inquiry Price
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SK&F 39728-A
T346523549-17-5
SK&F 39728-A is a bioactive chemical.
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Porcine dynorphin A(1-13)
TP117972957-38-1
Porcine dynorphin A (1-13) is a potent, endogenous κ opioid receptor agonist and is antinociceptive at physiological concentrations. Exposure to dynorphin A (1-13) causes acute increases in [Ca2+]i in individual neurons similar to increases seen with acut
  • $67
7-10 days
Size
QTY
1-[3’-O-[(4,4’-dimethoxytriphenyl)methyl]-a-L-threofuranosyl]-N6-benzoyladenine
TNU1629325683-88-3
1-[3’-O-[(4,4’-dimethoxytriphenyl)methyl]-a-L-threofuranosyl]-N6-benzoyladenine is a useful organic compound for research related to life sciences. The catalog number is TNU1629 and the CAS number is 325683-88-3.
  • Inquiry Price
7-10 days
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(R)-tert-Butyl (4-oxo-4-(3-(trifluoromethyl)-5,6-dihydro-[1,2,4]triazolo[4,3-a]pyrazin-7(8H)-yl)-1-(2,4,5-trifluorophenyl)butan-2-yl)carbamate
T65597486460-23-5
(R)-tert-Butyl (4-oxo-4-(3-(trifluoromethyl)-5,6-dihydro-[1,2,4]triazolo[4,3-a]pyrazin-7(8H)-yl)-1-(2,4,5-trifluorophenyl)butan-2-yl)carbamate is a useful organic compound for research related to life sciences and the catalog number is T65597.
    7-10 days
    Inquiry
    Amicoumacin A FA
    T23725L
    Amicoumacin A FA has antimicrobial activity, inhibiting S. purpureus and S. aureus, and can be used in the study of microbial infections.
    • $195
    In Stock
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    CCK-A receptor inhibitor 1
    T12404137004-80-9
    CCK-A receptor inhibitor 1 is a potent inhibitor of the cholecystokinin A (CCK-A) receptor (IC50: 340 nM).CCK-A receptor inhibitor 1 can be used for the study of diseases related to the digestive system.
    • $700
    6-8 weeks
    Size
    QTY
    Aurora A inhibitor 1
    T634362677799-04-9
    Aurora A inhibitor 1 is a potent and selective Aurora A inhibitor. Aurora A is associated with cancers of multiple histological origins and may exhibit oncogenic activity when overexpressed. aurora A inhibitor 1 exhibits potential for Aurora A-mediated cancer disease studies.
    • $2,140
    10-14 weeks
    Size
    QTY
    MAO A/HDAC-IN-1
    T61958
    MAO A/HDAC-IN-1 is an effective monoamine oxidase A (MAO A) and HDAC dual inhibitor, which can be used for glioma research.
    • $1,520
    10-14 weeks
    Size
    QTY
    1-Acetyltagitinin A
    TN252560547-63-9
    1-Acetyltagitinin A is a natural product of Tithonia, Asteraceae. The catalog number is TN2525 and the CAS number is 60547-63-9. 1-Acetyltagitinin A can be used as a reference standard.
    • $550
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    Aurora A/PKC-IN-1
    T629452143100-98-3
    Aurora A/PKC-IN-1 (Compound 2e) is a potent dual inhibitor of Aurora A (AurA) and PKC (α, β1, β2, θ), acting on AurA (IC50: 6.9 nM) and PKCα (IC50: 16.9 nM). Aurora A/PKC-IN-1 showed anti-proliferative and anti-metastatic effects on breast cancer cells.
    • $2,140
    6-8 weeks
    Size
    QTY
    Combretastatin A-1 phosphate tetrasodium
    T40367288847-34-7
    Combretastatin A-1 phosphate (OXi-4503) tetrasodium, a prodrug of Combretastatin A-1, is a tubulin-binding microtubule polymerization inhibitor that targets the colchicine-binding site. By inducing tubulin depolymerization, Combretastatin A-1 phosphate tetrasodium inhibits the Wnt/β-catenin pathway and leads to the deactivation of AKT. It possesses both anti-tumor and anti-vascular properties.
    • Inquiry Price
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    Dynorphin A (1-8)
    T2040375790-53-3
    Dynorphin (1-8) is an opioid octapeptide from the porcine hypothalamus. It comprises the N-terminal eight residues of dynorphin.
    • Inquiry Price
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    Lodenosine
    T19688110143-10-7
    Lodenosine is an inhibitor of RNA-directed DNA polymerase, and potentially for the treatment of HIV.
    • $1,520
    6-8 weeks
    Size
    QTY
    Prodilidine hydrochloride
    T284513734-16-5
    Prodilidine hydrochloride is an opioid analgesic.
    • $1,820
    8-10 weeks
    Size
    QTY